Books

G. Haufe and F. Leroux (Eds.), Fluorine in Life Sciences: Pharmaceuticals, Medicinal Diagnostics, and Agrochemicals, Academic Press, San Diego, 2019. (ISBN 978-0-12-812733-9)

A. Tressaud and G. Haufe (Eds.), Fluorine and Health. Molecular Imaging, Biomedical Materials and Pharmaceuticals, Elsevier, Amsterdam, 2008. (ISBN 978-0-444-53086-8)

G. Haufe and G. Mann, Chemistry of Alicyclic Compounds, Elsevier, Amsterdam, 1989. (ISBN 0-444-98878-5).

Publications

2023:

M. Essers and G. Haufe, „Synthesis of Diastereomeric 8-Fluoro-ABC-Steroid Building Blocks”, Eur. J. Org. Chem. 2023, e202300206. DOI

G. Haufe, „Selective Synthesis of Monofluorinated Compounds Applying Amine/HF Reagents”, Bioorg. Med. Chem. 2023, Chem. Rec. 2023, e202300140 (1-31). DOI

C. P. Konken, B. Beutel, B. Schinor, J. Song, H. Gerwien, E. Korpos, M. Burmeister, B. Riemann, M. Schäfers, L. Sorokin, and G. Haufe, „Influence of N-Arylsulfonamido D-Valine N-Substituents on the Selectivity and Potency of Matrix Metalloproteinase Inhibitors”, Bioorg. Med. Chem. 2023, 90, 117350. DOI

2022:

A. V. Chernyk, D. Alonsyn, Y. O. Kuchkovska, C. G. Daniliuc, N. A. Tolmachova, I. S. Kondratov, S. Zozula, O. O. Grygorenko, and G. Haufe, “Impact of β-perfluoroalkyl substitution of proline on the proteolytic stability of its amide derivatives”, Org. Biomol. Chem. 2022, 20, 9337-9350. DOI

P. Dudziński, A. V. Matsnev, J. S. Thrasher, and G. Haufe, “Reactions of difluoro-pentafluorosulfanyl-iodomethane (SF₅CF₂I) with electronically different types of alkenes”, J. Fluorine Chem. 2022, 264, 110051. DOI

I. Liashkovich, S. T. Stefanello, R. Vidyadharan, G. Haufe, A. Erofeev, P. V. Gorelkin, V. Kolmogorov, C. Rigon Mizdal, A. Dulebo, E. Bulk, I. U. Kouzel, and V. Shahin, “Pitstop-2 and its novel derivative RVD-127 disrupt global cell dynamics and nuclear pores integrity by direct interaction with small GTPases”, Bioengin. Transl. Med. 2022, e10425. DOI

I. G. Logvinenko, I. S. Kondratov, S. O. Pridma, N. A. Tolmachova, R. N. Morev, V. G. Dolovanyuk, C. Mück-Lichtenfeld, C. G. Daniliuc and G. Haufe, “Synthesis and physical chemical properties of CF₃O-containg secondary amines - perspective building blocks for drug discovery”, J. Fluorine Chem. 2022, 257-258, 109990. DOI

G. Haufe, “Synthesis and application of pentafluorosulfanylation reagents and aliphatic SF₅-containing building blocks”, Tetrahedron 2022, 109, 132656. DOI

L. Honold, M. Austrup, A. Faust, C. P. Konken, K. Schwegmann, B. Zinnhardt, C. G. Daniliuc, G. Haufe, M. Schäfers, K. Kopka, and S. Hermann, „Towards optimized bioavailability of ^99mTc-labeled barbiturates for non-invasive imaging of matrix metalloproteinase activity”, Mol. Imag. Biol. 2022, 24, 434-443. DOI

2021:

S. P. Belina, S.-Y. Qing, P. Dudziński, A. V. Matsnev, C. Mück-Lichtenfeld, G. Haufe, and J. S. Thrasher, “Preparation and Characterization of Pentafluoro-λ⁶-sulfanyldifluoromethane and Pentafluoro-λ⁶-sulfanyl-1,1,2,2-tetrafluoroethane”, Helv. Chim. Acta 2021, 104, e2100138. DOI

P. Dudziński, W. S. Husstedt, A. V. Matsnev, J. S. Thrasher, and G. Haufe, “Synthesis and [3,3]-sigmatropic rearrangements of (E)-5-(pentafluoro-λ⁶-sulfanyl)-pent-3-en-2-ol, its homologues and trifluoromethyl analogues”, Org. Biomol. Chem. 2021, 19, 5607-5623. DOI

2020:

E. N. Shaitanova, I. I. Gerus, O. A. Balabon, V. E. Ivasyshyn, K. V. Tarasenko, C. G. Daniliuc and G. Haufe, “Synthesis of fluorine-containing 3-aminocyclopent-2-enones via intramolecular cyclization”, Eur. J. Org. Chem. 2020, 7156-7163. DOI

B. Schinor, S. Hruschka, C. G. Daniliuc, D. Schepmann, B. Wünsch, and G. Haufe, “Fluorinated 2-Arylcyclopropan-1-amines – A New Class of Sigma Receptor Ligands”, Bioorg. Med. Chem. 2020, 28, 115726. DOI

I. O. Feskov, B. O. Golub, B. V. Vashchenko, V. V. Levterov, I. S. Kondratov, O. O. Grygorenko, and G. Haufe, “GABA analogues and related mono-/bifunctional building blocks derived from the fluorocyclobutane scaffold”, Eur. J. Org. Chem. 2020, 4755-4767. DOI

G. Haufe, “Pentafluorosulfanylation of Aliphatic Substrates”, Emerging Fluorinated Motifs: Synthesis, Properties and Applications, D. Cahard, J.-A. Ma, Eds., Wiley-VCH, Weinheim, 2020, Vol 2, pp 571-609. DOI

K. Schwegmann, M. Hohn, S. Hermann, M. Schäfers, B. Riemann, G. Haufe, S. Wagner, and H.-J. Breyholz, „Optimizing the biodistribution of radiofluorinated barbiturate tracers for MMP imaging by introduction of fluorescent dyes as pharmacokinetic modulators”, Bioconj. Chem. 2020, 31, 1117-1132. DOI

I. G. Logvinenko, Y. Markushyna, I. S. Kondratov, B. V. Vashenko, M. Kliachyna, Y. Tokaryeva, V. Pivnytska, O. O. Grygorenko, and G. Haufe, “Synthesis, physico-chemical properties and metabolic stability of compounds bearing aliphatic trifluoromethoxy group, J. Fluorine Chem. 2020, 231, 109461. DOI

V. Hugenberg, G. Haufe, “Fluorinated Matrix Metalloproteinase Inhibitors (MMPIs) for Potential Application in Therapy and Diagnosis of Diseases”, Frontiers of Organofluorine Chemistry, I. Ojima, Ed., World Scientific, London, 2020, pp 447-516. DOI

2019:

G. Haufe, “Synthesis of Fluoroalkanes by Addition Reactions to Alkenes”, Science of Synthesis, Fluorine, Vol. 34, Update 2019-3, Chapter 1.5, J.-F. Paquin, Ed., Thieme-Verlag, Stuttgart, 2019, 3, pp 141-332. DOI

G. Haufe, “Et3N∙3HF Complex Fluorination for Preparing Alkyl Fluorides, Synthetic Organofluorine Chemistry. Fluorination, J. Hu, T. Umemoto, Eds., Springer-Nature, Singapore, 2019, pp 1-44. DOI

2018:

B. Beutel, J. Song, C. P. Konken, E. Korpos, B. Schinor, H. Gerwien, R. Vidyadharan, M. Burmeister, L. Li, G. Haufe, and L. Sorokin, “Novel in vivo inhibitors for the matrix metalloproteinase (MMP)-2 and MMP-9”, Bioconj. Chem., 2018, 29, 3715-3725.DOI

M. Hohn, M. Chang, J. E. Meisel, E. Frost, K. Schweigmann, S. Hermann, M. Schäfers, B. Riemann, G. Haufe, H.-J. Breyholz, and S.Wagner, „Synthesis and preliminary in vitro and in vivo evaluation of thiirane-based slow binding MMP inhibitors as potential radiotracers for PET imaging”, ChemistrySelect, 2018, 3, 11729-11736.DOI

N. A. Tolmachova, I. S. Kondratov, V. G. Dolovanyuk, S. O. Pridma, A. V. Chernykh, C. G. Daniliuc and G. Haufe, “Synthesis of New fluorinated proline analogs from polyfluoroalkyl β-ketoacetals and ethyl isocyanoacetate”, Chem. Commun., 2018, 54, 9683-9687.DOI

V. Hugenberg, M. Behrends, S. Wagner, S. Hermann, M. Schäfers, H. C. Kolb, K. Szardenings, J. C. Walsh, L. F. Gomez, K. Kopka and G. Haufe, „Synthesis, radiosynthesis, in vitro and first in vivo evaluation of a new matrix metalloproteinase inhibitor based on γ-fluorinated α-sulfonylaminohydroxamic acid”, EJNMMI Radiopharm. Chem. 2018, 3(10), 1-20.DOI

I. S. Kondratov, N. A. Tolmachova, and G. Haufe, “Diels-Alder reaction in synthesis of fluorinated (hetero)aromatic compounds”, Eur. J. Org. Chem 2018, 14, 3618-3647.DOI

C. P. Konken, G. Haufe, K. Brömmel, B. Wünsch, M. Schäfers, S. Wagner and V. Hugenberg, “ Development of symmetric O-BODIPYs with different optical properties as building blocks for the synthesis of ligands for multimodal imaging”, Dyes & Pigments 2018, 158, 88–96.DOI

I. S. Kondratov, M. Y. Bugera, N. A. Tolmachova, C.-G. Daniliuc and G. Haufe, “Straightforward synthesis of fluorinated amino acids by Michael addition of ethyl bromodifluoroacetate to α,β-unsaturated α-amino acid derivatives”, J. Fluorine Chem. 2018, 211, 100-108.DOI

A.-L. Dreier, A. V. Matsnev, J. S. Thrasher, and G. Haufe, “Syn-selective silicon Mukaiyama-type aldol reactions of (pentafluoro-λ6-sulfanyl)acetic acid esters with aldehydes”, Beilstein J. Org. Chem. 2018, 14, 373–380.DOI

2017:

V. Kozel, P. Kirsch, C.-G. Daniliuc, and G. Haufe, „C3-symmetric tricyclo[2.2.1.0^2,6]heptane-3,5,7-triol”, Angew. Chem. Int. Ed. 2017, 56, 15456-15460.DOI; Angew. Chem. 2017, 129, 15659-15663.DOI
(Highlighted in Chem. Engin. News 2017, 95(46) 9 (Nov 20th, 2017).

I. O. Feskov, A. V. Chernykh, I. S. Kondratov, M. Klychina, C.-G. Daniliuc, and G. Haufe, „Cyclobutyl-containing rigid analogues of threonine: synthesis and physical chemical properties”, J. Org. Chem. 2017, 82, 12863-12868. DOI

K. Bartels, B. Schinor, and G. Haufe, “Diastereoselectivity of Cyclopropanation of Substituted α-Fluorostyrenes versus Styrenes by Different Methods”, J. Fluorine Chem. 2017, 203, 200-205.DOI

M. T. Borrello, B. Schinor, K. Bartels, H. Benelkebir, S. Pereira, W. T. Al-Jamal, L. R. Douglas, P. J. Duriez, G. K. Packham, G. Haufe, and A. Ganesan, “Fluorinated tranylcypromine analogues as inhibitors of lysine-specific demethylase 1 (LSD1, KDM1A)”, Bioorg. Med. Chem. Lett. 2017, 27, 2099-2101.(DOI)

C. P. Ortmayer, G. Haufe, K. Schwegmann, S. Hermann, M. Schäfers, F. Börgel, B. Wünsch, S. Wagner, and V. Hugenberg, “Synthesis and evaluation of a [¹⁸F]BODIPY-labeled Caspase-inhibitor”, Bioorg. Med. Chem. 2017, 25, 2167-1276.(DOI)

A.-L. Dreier, B. Beutel, C. Mück-Lichtenfeld, A. V. Matsnev, J. S. Thrasher, and G. Haufe, “The Ireland-Claisen rearrangement as a useful tool for the synthesis of new α-(pentafluorosulfanyl)- and α-(trifluoromethyl)-substituted carboxylic acid derivatives”, J. Org. Chem.. 2017, 82, 1638-1648.(DOI)

I. S. Kondratov, I. G. Logvinenko, N. A. Tolmachova, R. V. Morev, M. A. Kliachyna, F. Clausen, C. G. Daniliuk, and G. Haufe, “Synthesis and physical chemical properties of 2-amino-4-(trifluoromethoxy)butanoic acid - a CF₃O-containing analogue of natural lipophilic amino acids”, Org. Biomol. Chem. 2017, 15, 672-679.(DOI)

T. Borisova, N. Pozdnyakova, E. Shaitanova, I. Gerus, M. Dudarenko, G. Haufe, and V. Kukhar, “Effects of new fluorinated analogues of GABA, Pregabalin bioisosters, on the ambient level and exocytotic release of [³H]GABA from rat brain nerve terminals”, Bioorg. Med. Chem. 2017, 25, 759-764.(DOI)

2016:

A. V. Chernykh, I. O. Feskov, A. V. Chernykh, I. S. Kondratov, N. A. Tolmachova, D. S. Radchenko, C. G. Daniliuc, and G. Haufe, “ Synthesis and physical chemical properties of cis- and trans-1-amino-3-fluoro-3-methylcyclobutanecarboxylic acids”, Eur. J. Org. Chem. 2016, 4782-4786.(DOI)

J. Tanaka, S. Suzuki, E. Tokunaga, G. Haufe, and N. Shibata, „Asymmetric Desymmetrization via Non-metallic C-F Bond Activation: Synthesis of 3,5-Diaryl-5-fluoromethyl-oxazolidin-2-ones with Quaternary Carbon Center”, Angew. Chem. Int. Ed. . 2016, 55, 9432-9436.(DOI); Angew. Chem. 2016, 128, 9581-9586.(DOI)

D. Ulbrich, C.-G. Daniliuc, and G. Haufe, „Halofluorination of N-protected α,β-dehydro-α-amino acid esters – a convenient synthesis of α-fluoro-α-amino acid derivatives”, J. Fluorine Chem. 2016, 188, 65-75.(DOI)

P. Dudziński, A. V. Matsnev, J. S. Thrasher, and G. Haufe, „Synthesis of SF₅CF₂-Containing Enones and Instability of This Group in Specific Chemical Environments and Reaction Conditions”, J. Org. Chem. 2016, 81, 4454-4463.(DOI)

D. C. Ramb, A. Lerchen, M. Kischkewitz, B. Beutel, S. Fustero, and G. Haufe, „Addition of Nucleophiles to Fluorinated Michael Acceptors”, Eur. J. Org. Chem. 2016, 1751-1759.(DOI)

F. W. Friese, A.-L. Dreier, A. V. Matsnev, C.-G. Daniliuc, J. S. Thrasher, and G. Haufe, „Anti-selective Aldol Reactions of SF5-Acetic Acid Esters with Aldehydes Mediated by Dicyclohexylchloroborane”, Org. Lett. 2016, 18, 1012-1015.(DOI)

R. Lázaro, R. Román, D. M. Sedwick, G. Haufe, P. Barrio, and S. Fustero, „Asymmetric Synthesis of Monofluorinated 1-Amino-1,2-digydronaphthalene and 1,3-Aminoalkohol Derivatives”, Org. Lett. 2016, 18, 948-951.(DOI)

D. Ulbrich, C.-G. Daniliuc, and G. Haufe, „Synthesis of α,ω polyfluorinated α-amino acid derivatives and δ,δ difluoronorvaline”, Org. Biomol. Chem. 2016, 14, 2755-2767.(DOI)

B. Beutel, C. G. Daniliuc, B. Riemann, M. Schäfers, G. Haufe, „Fluorinated matrix metalloproteinases inhibitors - Phosphonate based potential probes for positron emission tomography”, Bioorg. Med. Chem. 2016, 24, 902-909.(DOI)

2015:

I. S. Kondratov, M. Ya. Bugera, N. A. Tolmachova, G. G. Posternak, C. G. Daniliuk, and G. Haufe, „Radical Reactions of Alkyl 2-Bromo-2,2-difluoroacetates with Vinyl Ethers: “Omitted” Examples and Application for the Synthesis of 3,3-Difluoro-GABA”, J. Org. Chem. 2015, 80, 12258-12264.(DOI)

R. S. Shaikh, P. Keul, M. Schäfers, B. Levkau, and G. Haufe, „New Fluorinated Agonists for Targeting the Sphingosin-1-Phosphate Receptor 1 (S1P1)”, Bioorg. Med. Chem. Lett. 2015, 25, 5048-5051.(DOI)

A. X. Chernykh, D. X. Radchenko, I. S. Kondratov, N. A. Tolmachova, O. X. Datsenko, M. A. Kurkunov, S. X. Zozulya, Y. X. Kheylik, K. Bartels, C. G. Daniliuk, and G. Haufe, „Synthesis and Physical-chemical Properties of 3-Fluorocyclobutyl Amines”, Eur. J. Org. Chem. 2015, 6466-6471.(DOI)

C. M. Waldmann, S. Hermann, A. Faust, B. Riemann, O. Schober, M. Schäfers, G. Haufe, and K. Kopka, „Novel fluorine-18 labeled 5-(1-pyrrolidinylsulfonyl)-7-azaisatin derivatives as potential PET tracers for in vivo imaging of activated caspases in apoptosis”, Bioorg. Med. Chem. 2015, 23, 5734-5739.(DOI)

T. Borisova, N. Pozdnyakova, E. Shaitanova, I. Gerus, M. Dudarenko, R. Mironets, G. Haufe, and V. Kukhar, “Synthesis of new fluorinated analogs of GABA, Pregabalin bioisosteres, and their effects on [H-3]GABA uptake by rat brain nerve terminals”, Bioorg. Med. Chem. 2015, 23, 4316-4323.(DOI)

P. Limpachayaporn, M. Schäfers, and G. Haufe,“Isatin Sulfonamides: Potent Caspases-3 and -7 Inhibitors and Potential PET and SPECT Radiotracers for Apoptosis Imaging”, Future Med. Chem. 2015, 7, 1173-1196.(DOI)

M. Behrends, S. Wagner, K. Kopka, S. Schröer, O. Schober, M. Schäfers, S. Kumbhar, M. Waller and G. Haufe,“New Matrix-Metallo-Proteinase Inhibitors Based on γ-Fluorinated α-aminocarboxylic and α-aminohydroxamic acids”, Bioorg. Med. Chem. 2015, 23, 3809-3818.(DOI)

N. Boechat, A. S. Carvalho, M. M. Bastos, K. Salomão, S. L. De Castro, C. F. Araujo-Lima, F. V. C. Mello, I. Felzenszwalb, C. Aiub, T. R. Condre, H. P. S. Zamith, R. Skupin and G. Haufe,“Studies of Genotoxicity and Mutagenicity of Nitroimidazoles: Demystifying this Critical Relationship with the Nitro Group”, Memórias do Instituto Oswaldo Cruz 2015, 110, 492-499.(DOI)

C. Nussbaum, S. Bannenberg, P. Keul, M. H. Gräler, C. F. Goncalves-De-Albuquerque, H. Korhonen, K. von Wnuk Lipinski, G. Heusch, H. C. F. Neto, I. Rohwedder, J. Göthert, V. P. Prasad, G. Haufe, B. Lange-Sperandio, S. Offermanns, M. Sperandio, and B. Levkau,“Sphingosin-1-phosphate receptor 3 promotes leukocyte rolling by mobilizing endothelial P-selectin”, Nature Commun. 2015, N°7416, 1-12.(DOI)

I. S. Kondratov, N. A. Tolmachova, V. G. Dolovanyuk, I. I. Gerus, C.-G. Daniliuk, and G. Haufe,“Synthesis of New Trifluoromethyl Containing Polysubstituted Aromatic Compounds by Diels-Alder Reaction of Ethyl 3-Benzamido-2-oxo-6-(trifluoromethyl)-2H-pyran-5-carboxylate”, Eur. J. Org. Chem. 2015, 2482-2491.(DOI)

R. S. Shaikh, S. S. Schilson, S. Wagner, S. Hermann, P. Keul, B. Levkau, M. Schäfers, and G. Haufe,“Synthesis and Evaluation of Fluorinated Fingolimod (FTY720) Analogues for Sphingosine-1-Phosphate Receptor Molecular Imaging by Positron Emission Tomography”, J. Med. Chem. 2015, 58, 3471-3484.(DOI)

P. Dudziński , A. Matsnev, J. S. Thrasher, and G. Haufe,"Ambiphilic Properties of SF₅CF₂CF₂Br Derived Perfluorinated Radical in Addition Reactions Across Carbon–Carbon Double Bonds", Org. Lett. 2015, 17, 1078–1081.(DOI)

S. S. Schilson, P. Keul, R. S. Shaikh, M. Schäfers, B. Levkau, and G. Haufe,“Synthesis of New Ligands for Targeting the S1P₁ Receptor”, Bioorg. Med. Chem. 2015, 23, 1011-1026.(DOI)

S. Fustero, A. Simón-Fuentes, P. Barrio, and G. Haufe,“Olefin Metathesis Reactions with Fluorinated Substrates, Catalysts and Solvents”, Chem. Rev. 2015, 115, 871-930.(DOI)

2014:

W. Alsibai, A. Hanenkamp, M. Eisenblätter, B. Riemann, M. Schäfers, C. Bremer, G. Haufe, and C. Höltke,“Fluorescent Non-peptidic RGD Mimetics with High Selectivity for αvβ3 vs αIIbβ3 Integrin Receptors: Novel Probes for in Vivo Optical Imaging”, J. Med. Chem. 2014, 57, 9971-9982.(DOI)

P. Limpachayaporn, S. Wagner, K. Kopka, O. Schober, M. Schäfers, and G. Haufe,“Novel 7-Halogenated Isatin Sulfonamides: Metabolically More Stable Inhibitors of Caspase-3 and -7 and Potential PET and SPECT Imaging Agents for Apoptosis”, J. Med. Chem. 2014, 57, 9383-9395.(DOI)

M. Marhold, C. Stillig, R. Fröhlich, G. Haufe,“Ring-Closing Metathesis of Vinyl Fluorides towards α-Fluorinated α,ß-Unsaturated Lactams and Lactones”, Eur. J. Org. Chem. 2014, 5777-5785.(DOI)

A.-L. Dreier, A. V. Matsnev, J. S. Thrasher, G. Haufe,“New approach to α-pentafluorosulfanyl-substituted carboxylic acid derivatives via Ireland-Claisen rearrangements”, J. Fluorine Chem. 2014, 167, 84-90.(DOI)

V. P. Prasad, S. Wagner, P. Keul, S. Hermann, B. Levkau, M. Schäfers, G. Haufe,“Synthesis of fluorinated analogues of sphingosine-1-phosphate antagonists as potential radiotracers for molecular imaging using positron emission tomography”, Bioorg. Med. Chem. 2014, 22, 5168-5181.(DOI)

D. C. Ramb, L. Kost, and G. Haufe, “[3,3]-Sigmatropic rearrangements of fluorinated allyl (thio)cyanates – tool for the synthesis of fluorinated (thio)ureas”, Chimia 2014, 68, 436-441.(DOI)

A. V. Matsnev, S.-Y. Qing, M. A. Stanton, K. A. Berger, G. Haufe, and J. S. Thrasher, “Pentafluorosulfanyldifluoroacetic acid – rebirth of a promising building-block”, Org. Lett. 2014, 16, 2402-2405.(DOI)

I. S. Kondratov, N. A. Tolmachova, V. G. Dolovanyuk, I. I. Gerus, K. Bergander, C.-G. Daniliuc, and G. Haufe, “Diels-Alder reaction of ethyl 3-benzamido-2-oxo-6-(trifluoromethyl)-2H-pyran-5-carboxylate with alkoxyalkenes as an effective approach to new trifluoromethyl containing 3-aminobenzoic acid derivatives”, Eur. J. Org. Chem. 2014, 2443-2450.(DOI)

U. I. M. Gerling, M. Salwiczek, C. D. Cadikamo, H. Erdbrink, S. L. Grage, P. Wadwani, A. S. Ulrich, M. Behrends, G. Haufe, C. Czekelius and B. Koksch, "Partial side chain fluorination influencing amyloid formation: a systematic study including size, hydrophobicity, and α-helix propensity“, Chem. Sci. 2014, 5, 819-830.(DOI)

E. N. Shaitanova, I. I. Gerus, V. P. Kukhar and G. Haufe, "Synthesis of enantiopure diastereomers of 4-Polyfluoromethyl-4-hydroxy Homoprolines by intramolecular cyclization of ε-aminoacrylic acids“, J. Fluorine Chem. 2014, 160, 8-11.(DOI)

2013:

S. Fustero, P. Bello, J. Miró, M. Sánchez-Rosello, G. Haufe and C. del Pozo, "One pot Cross Enyne Metathesis (CEYM) - Diels Alder Reaction of gem-Difluoropropargylic Alkynes“, Beilstein J. Org. Chem. 2013, 9, 2688-2695.(DOI)

Daniel C. Ramb and G. Haufe, "Overman rearrangement of fluorinated allylic alcohols as a key step for the synthesis of glycyldecylamide (GDA) mimics“, Synlett 2013, 24, 2229-2232.(DOI)

B. Schinor, B. Wibbeling, and G. Haufe, "Synthesis and pKa values of 2-3- and 4-pentafluorosulfanyl-phenyl)-2-fluorocyclopropylamines", J. Fluorine Chem. 2013, 155, 102-109.(DOI)

P. Limpachayapron, S. Wagner, K. Kopka, S. Hermann, M. Schäfers and G. Haufe, "Synthesis, [¹⁸F]-Radiolabeling and in vivo Biodistribution Studies of N-Fluorohydroxybutyl Isatin Sulfonamides for Apoptosis Imaging using Positron Emission Tomography (PET)", J. Med. Chem. 2013, 56, 4509-4520.(DOI)

C. Waldmann, O. Schober, G. Haufe and K. Kopka, A Closer Look at the Bromine-Lithium Exchange with tert-Butyllithium within a Synthesis of Aryl Sulfonamides, Org. Lett. 2013, 15(12), 2954-2957.(DOI)

M. Lübke, M. Jung and G. Haufe, "New Histone Deacetylase Inhibitors based on 2-Amino-4-fluorocarboxylic Acid Esters: Synthesis and Activity", J. Fluorine Chem. 2013, 152, 144-156.(DOI)

I. P. Limpachayaporn, B. Riemann, K. Kopka, O. Schober, M. Schäfers and G. Haufe, "Influence of 4- or 5-Substituents on the Pyrrolidine Ring of 5-[1-(2-Methoxymethylpyrrolidinyl)sulfonyl]isatin Derivatives on Their Inhibitory Activities towards Caspases-3 and -7", Eur. J. Med. Chem. 2013, 64, 562-578.(DOI)

P. Limpachayaporn, M. Schäfers, O. Schober, K. Kopka and G. Haufe, "Synthesis of New Fluorinated, 2-Substituted 5-Pyrrolidinylsulfonyl Isatin Derivatives as Caspase-3 and Caspase-7 Inhibitors: Nonradioactive Counterparts of Putative PET-compatible Apoptosis Imaging Agents", Bioorg. Med. Chem. 2013, 21, 2025-2036.(DOI)

2012:

G. Haufe, "Putting a Greenhouse Gas to Work", Science 2012, 338, 1298-1298.

G. Haufe, S. Suzuki, H. Yasui, C. Terada, T. Kitayama, M. Shiro and N. Shibata, "C-F Bond Activation of Non-activated Aliphatic Fluorides: Synthesis of Fluoromethyl-3,5-diaryl-2-oxazolidinones by Desymmetrization of 2-Aryl-1,3-difluoropropan-2-ols", Angew. Chem. 2012, 124, 12441-12445; Angew. Chem. Int. Ed. 2012, 51, 12275-12279.

P. Persich, J. Kerschbaumer, S. Helling, B. Hildmann, B. Wibbeling and G. Haufe, "Reactions of Transannular O-Heterocyclization: A Useful Tool for the Total Synthesis of Murisolin and 16,19-cis-Murisolin", Org. Lett. 2012, 14, 5628-5631.

I. S. Kondratov, V. G. Dolovanyuk, N. A. Tolmacheva, I. I. Gerus, K. Bergander, R. Fröhlich and G. Haufe, "Reactions of ß-Alkoxyvinyl Polyfluoroalkyl Ketones with Ethyl Isocyanoacetate and Its Use for the Synthesis of New Polyfluoroalkyl Pyrroles", Org. Biomol. Chem. 2012, 10, 8778-8785.

V. Hugenberg and G. Haufe, "Fluoro-Pummerer Rearrangement and Analogous Reactions", J. Fluorine Chem. 2012, 143, 238-262.

J. Walkowiak, H. Koroniak and G. Haufe, "Selectively Fluorinated Amides via Eschenmoser-Claisen-Type Rearrangement", J. Fluorine Chem. 2012, 143, 189-197.

D. Schrigten, H.-J. Breyholz, S. Wagner, S. Hermann, O. Schober, M. Schäfers, G. Haufe and K. Kopka, "A New Generation of Radiofluorinated Pyrimidine-2,4,6-triones as MMP-targeted Radiotracers for Positron Emission Tomography", J. Med. Chem. 2012, 55, 223-232.

I. Humelnicu, E.-U. Würthwein and G. Haufe, "The conformers of 3-Fluoroalanine. A Theoretical Study", Org. Biomol. Chem. 2012, 10, 2084-2093.

2011:

V. M. Muzalevskiy, A. V. Shastin, E. S. Balenkova, G. Haufe and V. G. Nenajdenko, "Synthesis of a-trifluoromethyl-phenethylamines from a-trifluoromethyl ß-aryl enamines and ß-chloro-ß-(trifluoromethyl)styrenes", J. Fluorine Chem. 2011, 132, 1247-1253.

J. Leuger, G. Blond, T. Billard, G. Haufe and B. R. Langlois, “1,4-Addition of Electron-rich Heterocycles onto β-Perfluoroalkyl Enones”, J. Fluorine Chem. 2011, 132, 799-803.

W. S. Husstedt, J. S. Thrasher and G. Haufe, „Synthesis of Pentafluorosulfany-1,3-Dienes”, Synlett 2011, 1683-1686.

N. A. Tolmachova, V. G. Dolovanyuk, I. I. Gerus, I. S. Kondrakov, V. V. Polovinko, K. Bergander and G. Haufe, „Catalytic Hydrogenation of 3-Amino-6-trifluoromethyl-pyridones and Its Use for the Synthesis of CF3-containing Mimetics of Ornithine and Thalidomide”, Synthesis 2011, 1149-1156.

W. S. Husstedt, S. Wiehle, C. Stillig, K. Bergander, S. Grimme and G. Haufe, „Synthesis and Preferred Conformations of All Regio- and Diastereoisomeric Methyl 2,3-Fluorohydroxyalkanoates”, Eur. J. Org. Chem. 2011, 355-363.

2010:

V. Hugenberg, R. Fröhlich and G. Haufe, “Oxidative desulfurization–fluorination of thioethers. Application for the synthesis of fluorinated nitrogen containing building blocks”, Org. Biomol. Chem. 2010, 8, 5682-5691.

V. Hugenberg, S. Wagner, K. Kopka, O. Schober, M. Schäfers and G. Haufe, „Synthesis of geminal difluorides by oxidative desulfurization-difluorination of alkyl aryl thioethers with halonium electrophiles in the presence of fluorinating reagents and its application for 18F-radiolabelling”, J. Org. Chem. 2010, 75, 6086-6095.

K. Koroniak and G. Haufe, „Synthesis of Enantiopure Fluorinated Ceramides; Analogues of Natural Sphingolipids”, Synthesis 2010, 75, 3309-3314.

V. Hugenberg and G. Haufe, „Facile Synthesis of a,a-Difluoroalkyl Aryl Thioethers and Their Oxidative Desulfurization-Fluorination to Trifluorides”, J. Fluorine Chem. 2010, 131, 942-950.

N. Purkayastha and G. Haufe, „An Efficient Access to Conformationally Rigid Amino Acid Analogues with a Piperidine Skeleton”, Synlett 2010, 1501-1504.

K. Koroniak and G. Haufe, „Stereoselective Synthesis of Fluorinated and Non-fluorinated Triazolo Analogues of Ceramides”, Synthesis 2010, 75, 498-504.

A. Y. Rulev, V. M. Muzalevskiy, E. V. Kondrashov, I. A. Ushakov, A. V. Shastin, E. S. Balenkova, G. Haufe, and V. G. Nenajdenko, „A Cascade Approach to Captodative Trifluorometrhylated Enamines or Vinylogous Guanidinium Salts: The Aromatic Substituent as a Switch of the Reaction Direction”, Eur. J. Org. Chem. 2010, 300-310.

N. Purkayastha, D. M. Shendage, and G. Haufe, „The Vinylfluoro Group as an Acetoyl Cation Equivalent. Stereoselective Synthesis of 6-Substituted 4-Hydroxy Pipecolic Acid Derivatives”, J. Org. Chem. 2010, 75, 222-225.

2009:

A. Faust, S. Hermann, S. Wagner, G. Haufe, O. Schober, M. Schäfers, and K. Kopka, „Molecular Imaging of Apoptosis in vivo with Scintigraphic and Optical Biomarkers - A Status Report”, Anti-Cancer Agents Med. Chem. 2009, 9, 968-985.

V. M. Muzalevskiy, A. V. Shastin, E. S. Balenkova, G. Haufe, and V. G. Nenajdenko, „Synthesis of Trifluoromethyl Pyrroles and Their Benzoanalogues”, Synthesis 2009, 3905-3929.

V. M. Muzalevskiy, V. G. Nenajdenko, A. V. Shastin, E. S. Balenkova, and G. Haufe, „Synthetic approach to alkoxy-β-(trifluoromethyl)styrenes and their application in synthesis of new trifluoromethylated heterocycles”, Synthesis 2009, 2249-2259.

A. K. Podichetty, S. Wagner, S. Schröer, A. Faust, O. Schober, M. Schäfers, K. Kopka, and G. Haufe, „Fluorinated isatin derivatives. Part 2. New N-substitutred 5-pyrrolidinylsulfonyl isatins as potential tools for molecular imaging of caspases in apoptosis”, J. Med. Chem. 2009,52, 3484-3495.

V. M. Muzalevskiy, V. G. Nenajdenko, A. Yu. Rulev, I. A. Ushakov, G. V. Romanenko, A. V. Shastin, E. S. Balenkova, and G. Haufe”, Selective synthesis of α-trifluoromethyl-β-aryl enamines or vinylogous guanidinium salts by treatment of β-halo-β-trifluoromethylstyrenes with secondary amines under different conditions”, Tetrahedron 2009, 65, 6991-7000.

A. K. Podichetty, S. Wagner, A. Faust, M. Schäfers, O. Schober, K. Kopka, and G. Haufe, „Fluorinated isatin derivatives. Part 3. New side-chain fluoro-functionalized pyrrolidinyl sulfonyl isatins as potent caspase-3 and –7 inhibitors”, Future Med. Chem. 2009, 1, 969-989.

V. M. Muzalevskiy, V. G. Nenajdenko, A. V. Shastin, E. S. Balenkova, and G. Haufe, “Synthesis of 1-trifluoromethyl-2-arylenamines and their untility for the Fischer indol synthesis and Pictet-Spengler reaction”, Tetrahedron 2009, 65, 7553-7561.

N. A. Tolmacheva, I. I. Gerus, V. G. Dolovanyuk, I. S. Kondratov, and G. Haufe, “Synthesis of new δ-(polyfluoroalkyl)-δ-hydroxy-α-amino acids”, Eur. J. Org. Chem. 2009, 5012-5019.

A. K. Podichetty, A. Faust, K. Kopka, S. Wagner, O. Schober, M. Schäfers and G. Haufe, "Fluorinated Isatin Derivatives. Paert 1. Synthesis of New N-Substituted (S)-5-[1-(2-Methoxymethylpyrrolidinyl)sulfonyl]isatins as Potent Caspase-3- and –7 Inhibitors", Bioorg. Med. Chem. 2009, 17, 2680-2688.

V. Hugenberg and G. Haufe, “Oxidative Desulfurization-Difluorination of Alkyl Aryl Thioethers: Synthesis of ?-Substituted 1,1-Difluoroalkanes”, Synlett 2009, 106-108.

2008:

V. N. Kovtonyuk, L. S. Kobrina, and G. Haufe, "Pentafluorophenylation of aromatic compounds with 4,5,6,7,8-pentafluoro-6-nitro-1-oxaspiro[2.5]octa-4,7-diene", Izv. Akad. Nauk, Ser. Khim. 2008, 57, 1654-1656; Russ. Chem. Bull. 2008, 57, 1686-1688.

V. M. Muzalevskiy, A. V. Shastin, E. S. Balenkova, G. Haufe, and V. G. Nenajdenko, „Novel Synthetic Pathway to 2-Trifluoromethylindole and 2-Amino-3-(trifluoromethyl)quinoline”, Izv. Akad. Nauk, Ser. Khim. 2008, 57, 2175-2177; Russ. Chem. Bull. 2008, 57, 2217-2219.

T. Billard, B. R. Langlois, M. Essers and G. Haufe, “Use of Cyclic α,β-Unsaturated Trifluoromethyl Sulfones in Diels-Alder Reactions and Michael Additions”, Collect. Czech. Chem. Commun. 2008, 73, 1814-1824.

I. Hyla-Kryspin, S. Grimme, S. Hruschka and G. Haufe, “Conformational Preferences and Basicities of Monofluorinated Cyclopropyl Amines in Comparison to Cyclopropylamine and 2-Fluoroethylamine”, Org. Biomol. Chem. 2008, 6, 4167-4175.

V. M. Muzalevskiy, V. G. Nenajdenko, A. V. Shastin, E. S. Balenkova, and G. Haufe, “Synthesis of Trifluoromethyl Alcohols from tert-Butoxy-β-(trifluoromethyl)styrenes and Trifluoromethylbenzyl ketones under the conditions of the Leuckart-Wallach Reaction”, J. Fluorine Chem. 2008, 129, 1052-1055.

V. M. Muzalevskiy, V. G. Nenajdenko, A. V. Shastin, E. S. Balenkova, and G. Haufe, “Application of 1-(3-Bromo-3,3-difluoroprop-1-ynyl)benzenes in Diels-Alder Reactions: Synthesis of ortho-CF2B-substituted Biaryls”, Synthesis, 2008, 2899-2904.

S. Hruschka, S. Yoshida, K. L. Kirk and G. Haufe, „Fluorinated Phenylcyclopropyl-amines. Part 6: Effects of Electron Withdrawing and Donating Aryl Substituents on the Inhibition of Tyramine Oxidase from Arthrobacter sp. by Diastereomeric 1-Aryl-2-fluoro-cyclopropylamines”, J. Fluorine Chem. 2008, 129, 875-880.

A. V. Shastin, V. G. Nenajdenko, V. M. Muzalevskiy, E. S. Balenkova, R. Fröhlich and G. Haufe, „New Synthetic Approach to a-Fluoro-ß-arylvinyl sulfones and Their Application in Diels-Alder Reactions”, Tetrahedron 2008, 64, 9725-9732.

S. Hruschka, T. C. Rosen, S. Yoshida, K. L. Kirk, R. Fröhlich, B. Wibbeling and G. Haufe, „Fluorinated Phenylcyclopropylamines. Part 5: Effects of Electron Withdrawing and Donating Aryl Substituents on the Inhibition of Monoamine Oxidases by 1-Aryl-2-fluoro -cyclopropylamines”, Bioorg. Med. Chem. 2008, 16, 7148-7166.

G. S. Nikolova and G. Haufe, “Stereoselective synthesis of (2S,3S)-4-fluoro-1,3-dihydroxy-2-octadecanoylamino-octadec-(4Z)-ene, [(Z)-4-fluoroceramide], and its phase behavior at the air/water interface”, Beilstein J. Org. Chem. 2008, 4, 12.

I. Hyla-Kryspin, G. Haufe and S. Grimme, “MP2 and QCISD(T) Study on the Convergence of Interaction Energies of Weak O-H•••F-C, C-H•••O, and C-H•••F-C Hydrogen Bridges”, Chem. Phys. 2008, 346, 224-236.

G. S. Nikolova, L. Zhang, X. Chen, L. Chi, and G. Haufe, „Selective Synthesis and Self-organization at the Air/Water Interface of Long Chain Fluorinated Unsaturated Ethyl Esters and Alcohols”, Colloids & Surfaces A: Physical and Engineering Aspects 2008, 317, 414-420 .

G. S. Nikolova and G. Haufe, “Selective Synthesis of Diastereomeric Fluorinated Octadeca-2,4-dienoic Acid Esters and Octadeca-2,4-dienols”, Synthesis 2008, 527-536.

K. L. Kirk, S. Yoshida and G. Haufe, “Synthesis and Biochemical Evaluation of Fluorinated Monoamine Oxidase Inhibitors”, Fluorine and Health: Molecular Imaging, Biomedical Materials and Pharmaceuticals, A. Tressaud, G. Haufe, Eds., Elsevier, Amsterdam, 2008, pp 659-695.

K. Kopka, S. Wagner, M. Schäfers, A. Faust, O. Schober and G. Haufe, “18F-labelled PET-Tracers for Cardiological Imaging”, Fluorine and Health: Molecular Imaging, Biomedical Materials and Pharmaceuticals , A. Tressaud, G. Haufe, Eds., Elsevier, Amsterdam, 2008, pp 85-139.

2007:

N. A. Tolmachova, I. I. Gerus, S. I. Vdovenko, G. Haufe and Y. A. Kizhner, “Synthesis of New Polyfluoroalkyl-containing Pyrones, Pyridones and Pyrido[1,2- a ]-benzazoles from Fluorinated ß-Alkoxyenones”, Synthesis 2007, 3797-3806.

S. Wagner, H.-J. Breyholz, M. P. Law, A. Faust, C. Höltke, S. Schröer, G. Haufe, B. Levkau, O. Schober, M. Schäfers and K. Kopka, „Novel fluorinated derivatives of the broad-spectrum MMP inhibitors N-Hydroxy-2(R)-[[4-methooxypenyl)sulfonyl](benzyl)- and (3-picolyl)-amino]3-methyl-butanamide (CGS 25966 and CGS 27023A) as a potential tool for the molecular imaging of activated MMPs with PET”, J. Med. Chem. 2007, 50, 5752-5764.

M. Marhold, U. Wittmann, S. Grimme, T. Takahashi, G. Haufe, „Synthesis of optically active 2-fluoroalk-1-en-3-yl esters and chirality transfer in their Claisen-type rearrangements”, J. Fluorine Chem. 2007, 128, 1306-1317.

J. Hajduch, O. Paleta, J. Kvícala and G. Haufe, „Fluorinated Furan-2(5H)-ones: Reactivity and Stereoselectivity in Diels-Alder Reactions”, Eur. J. Org. Chem. 2007, 5101-5111.

V. G. Nenajdenko, V. M. Muzalevskij, A. V. Shastin, E. S. Balenkova and G. Haufe, „Synthesis and Diels-Alder reactions of a-fluoro- and a-trifluoromethylacrylonitriles”, J. Fluorine Chem. 2007, 128, 818-826.

S. Steffens, U. Höweler, R. Rudert, J. Oldendorf, G. Haufe and H.-J. Galla, “Temperature Dependent Phase Behaviour and the Nucleation Process of Ethyl 4-Fluoro-2,3-dihydroxystearate Monolayers”, Langmuir 2007, 23, 1880-1887.

E. V. Panteleeva, G. Haufe and V. D. Shteingarts, „Short Access to 4-Alkenylbenzonitriles. Reaction of Anionic Reduced Forms of Terephthalonitrile with Alkenyl Bromides”, Synlett, 2007, 1616-1618.

S. Hruschka, R. Fröhlich, P. Kirsch and G. Haufe, „Synthesis of New Enantiopure Fluorinated Phenylcyclopropanecarboxylates. Potent Chiral Dopants for Liquid Crystal Compositions”, Eur. J. Org. Chem. 2007, 141-148.

M. Essers and G. Haufe, “ Tetrafluoro-p-benzoquinone in Synthesis”, in Encyclopedia of Reagents for Organic Synthesis L. A. Paquette, Ed., John Wiley & Sons, Inc., Chichester, 2007, 468-474, (electronic version , DOI: 10.1002/047084289X.rn00532, pp 1-13).

M. Essers and G. Haufe, “ Hexafluoro-2-butyne in Synthesis”, in Encyclopedia of Reagents for Organic Synthesis L. A. Paquette, Ed., John Wiley & Sons, Inc., Chichester, 2007, 295-304, (electronic version , DOI: 10.1002/047084289X.rn00624, pp 1-19).

M. Essers and G. Haufe, “ Difluoromaleic anhydride in Synthesis”, in Encyclopedia of Reagents for Organic Synthesis L. A. Paquette, Ed., John Wiley & Sons, Inc., Chichester, 2007, 206-207, (electronic version , DOI: 10.1002/047084289X.rn00623, pp 1-3).

M. Essers and G. Haufe, “ Difluoromaleic acid in Synthesis”, in Encyclopedia of Reagents for Organic Synthesis L. A. Paquette, Ed., John Wiley & Sons, Inc., Chichester, 2007, 204-205, (electronic version , DOI: 10.1002/047084289X.rn00622, pp 1-4).

M. Essers and G. Haufe, “2,6- Difluoro- p -benzoquinone in Synthesis”, in Encyclopedia of Reagents for Organic Synthesis L. A. Paquette, Ed., John Wiley & Sons, Inc., Chichester, 2007, 204 ( electronic version , DOI: 10.1002/047084289X.rn00533, pp 1-2).

M. Essers and G. Haufe, “2,3- Difluoro- p -benzoquinone in Synthesis”, in Encyclopedia of Reagents for Organic Synthesis L. A. Paquette, Ed., John Wiley & Sons, Inc., Chichester, 2007, 203 ( electronic version , DOI: 10.1002/047084289X.rn00534, pp 1-2).

2006:

P. Kirsch, A. Hahn, R. Fröhlich, G. Haufe, „Liquid Crystals Based on Axially Fluorinated 1,3-Dioxanes: Synthesis, Properties and Computational Study", Eur. J. Org. Chem. 2006, 4819-4824.

N. A. Tolmachova, I. I. Gerus, M. S. I. Vdovenko, M. Essers, R. Fröhlich and G. Haufe, „Thermal Diels-Alder Reactions of 3-(Benzoylamino)-6-(polyfluoroalkyl)pyran-2-ones - New Synthesis of p-(Polyfluoroalkyl)-anilines”, Eur. J. Org. Chem. 2006, 4704-4709.

F. Chanteau, R. Platier-Royong, G. Haufe and C. Portella, "Synthesis of o-Perfluoroalkyl Phenones from Hemifluorinated Enones as Key Building Blocks", Tetrahedron 2006, 62, 9049-9053.

J. Oldendorf and G. Haufe, "Synthesis of Both Enantiomers of the Diastereomeric 4-Fluoro Analogues of 4,5-Dihydroceramide", Eur. J. Org. Chem. 2006, 4463-4472.

U. Wittmann, F. Tranel, R. Fröhlich and G. Haufe, “ Novel Synthesis of 4-Fluoropyridines Based on 2-Fluoroallylic Alcohols by Succeeding Ireland-Claisen and Aza-Cope Rearrangements as Key Steps”, Synthesis 2006, 2085-2096.

J. Leuger, G. Blond, R. Fröhlich, T. Billard, G. Haufe and B. Langlois, “ Synthetic Application of ß-Fluoro-alkylated Enones. 1. Use as Dienophiles in Diels-Alder Cycloadditions”, J. Org. Chem. 2006, 71, 2735-2739.

S. Steffens, J. Oldendorf, G. Haufe, and H.-J. Galla, “Organized Collapse Structures in Mixtures of Chiral Ethyl 2-Azido-4-fluoro-3-hydroxystearates”, Langmuir 2006, 22, 1428-1435.

R. Fröhlich, T. C. Rosen, O. G. J. Meyer, K. Rissanen and G. Haufe, “New Indications for the Potential Involvement of C-F Bonds in Hydrogen Bonding”, J. Mol. Struct. 2006, 787, 50-62.

G. Haufe, “Synthesis of ß-Fluoroalkohols by Ring Opening of Epoxides, in Science of Synthesis , Vol 34, J. Percy (Ed.), Chapter 9.1, Thieme, Stuttgart, 2006, pp 345-378.

G. Haufe, “Synthesis of Halofluoroalkanes and Analogues by Addition Reactions to Alkenes, in Science of Synthesis , Vol 34, J. Percy (Ed.), Chapter 1.5, Thieme, Stuttgart, 2006, 169-223.

2005:

X. Chen, S. Wiehle, M. Weygand, G. Brezesinski, U. Klenz, H-J. Galla, H. Fuchs, G. Haufe, and L. Chi, "Unconventional Air-stable Interdigitated Bilayer Formed by 2,3-Disubstituted Fatty Acid Methyl Esters", J. Phys. Chem. B. 2005, 109, 19866-19875.

F. Tranel, R. Fröhlich and G. Haufe, "Synthesis of g-Fluoro-a-amino Acids by Claisen Rearrangement", J. Fluorine Chem. 2005, 126, 557-569.

I. I. Gerus, N. A. Tolmachova, S. I. Vdovenko, R. Fröhlich and G. Haufe, "A Convenient Synthesis and Chemical Properties of 3-Acylamino-6-polyfluoroalkyl-2H-pyran-2-ones", Synthesis 2005, 1269-1278.

X. Chen, S. Wiehle, L. Chi, C. Mück-Lichtenfeld, R. Rudert, D. Vollhardt, H. Fuchs, and G. Haufe, "Phase Behaviour of 2,3-Disubstituted Methyl Octadecanoate Monolayers at the Air-Water Interface", Langmuir 2005, 21, 3376-3383.

G. Haufe, "Vinyl Fluorides in Cycloadditions", in Fluorine-Containing Synthons, ACS Symposium Series, Vol. 911, Soloshonok, V. A., Ed., American Chemical Society, Washington, D.C., 2005, Chapter 7, pp 155-172.

V. N. Kovtonyuk, L. S. Kobrina, O. M. Katayeve and G. Haufe, "Reactions of Polyfluorinated Cyclohexadienones with Diazoalkanes. Part 2. Formation of Cyclohexadiene-spiro-Oxiranes from Polyfluorinated Cyclohexa-2,5-dienones with Diazomethane and Its Reactions with Aryl- and Chloroethyl Isocyanates", Eur. J. Org. Chem. 2005, 1178-1183.

S. Ye, S. Yoshida, R. Fröhlich, G. Haufe and K. Kirk, "Fluorinated Phenylcyclopropylamines: Part 4. Effects of Aryl Substituents and of Stereochemistry on the Inhibition of Monoamine Oxidase A and B by 1-Aryl-2-fluorocyclopropylamines", Bioorg. Med. Chem. 2005, 13, 2489-2499.

D. M. Shendage, R. Fröhlich, K. Bergander and G. Haufe, "Asymmetric Synthesis of g-Fluorinated a-Amino Acids", Eur. J. Org. Chem. 2005, 719-727.

2004:

T. C. Rosen, S. Yoshida, K. L. Kirk and G. Haufe, "Fluorinated Phenylcyclopropylamines: Part 2. Effects of Aromatic Ring Substitution and of Absolute Configuration on Inhibition of Microbial Tyramine Oxidase", J. Med. Chem. 2004, 47, 5860-5871.

D. M. Shendage, R. Fröhlich and G. Haufe, "Highly Efficient Stereo Conservative Amidation and Deamidation of g-Amino Acids", Org. Lett. 2004, 6, 3675-3678.

J. Walkowiak, G. Haufe and H. Koroniak, "New Application of 1,1,3,3,3-Pentafluoropropyl-diethylamine Adduct (PFPDEA) as Fluorinating Agent. Synthesis of 3,3,3-Trifluoropropionates of Vicinal Fluorohydrins", Polish J. Chem. 2004, 78, 1777-1784.

S. Behr, K. Hegemann, H. Schimanski, R. Fröhlich and G. Haufe, "Synthesis of g-Lactones from Cycloocta-1,5-diene - Starting Materials for Natural Product Synthesis", Eur. J. Org. Chem. 2004, 3884-3892.

F. Tranel and G. Haufe, "Claisen rearrengments based on vinyl fluorides", J. Fluorine Chem.. 2004, 125, 1593-1608.

I. Hyla-Kryspin, G. Haufe and S. Grimme, "Weak Hydrogen Bridges: A Systematic Theoretical Study on the Nature and Strength of C-H···F-C Interactions", Chem. Eur. J. 2004, 10, 3411-3422.

T. C. Rosen, S. Yoshida, K. L. Kirk and G. Haufe, "Fluorinated Phenylcyclopropylamines as Inhibitors of Monoamine Oxidases", ChemBioChem. 2004, 5, 1033-1043.

G. Haufe, "Regio- and Stereoselective Synthesis of Vicinal Fluorohydrins", J. Fluorine Chem. 2004, 125, 875-894.

S. Yoshida, T. C. Rosen, O. G. J. Meyer, S. Ye, M. J. Sloan, G. Haufe and K. L. Kirk, “Fluorinated Phenylcyclopropylamines: Part 3. Inhibition of Monoamine Oxidases A and B”, Biorg. Med. Chem. 2004, 12, 2645-2652.

K. Hegemann, R. Fröhlich and G. Haufe, “Synthesis of Enantiopure 9-Oxabicyclononanediol Derivatives by Lipase-catalyzed Transformations”, Eur. J. Org. Chem. 2004, 2181-2192.

S. Yoshida, O. G. J. Meyer, T. C. Rosen, G. Haufe S. Ye, M. J. Sloan and K. L. Kirk, “Fluorinated Phenylcyclopropylamines: Part 1. Synthesis and Effect of Fluorine Substitution at the Cyclopropane Ring on Inhibition of Microbial Tyramine Oxidase”, J. Med. Chem. 2004, 47, 1796-1806.

T. C. Rosen, E. De Clercq, J. Balzarini and G. Haufe, “Synthesis and Antiviral Activity of Monofluorinated Cyclopropanoid Nucleosides”, Org. Biomolec. Chem. 2004, 2, 229-237.

M. Marhold, A. Buer, H. Hiemstra, J. H. van Maarseveen and G. Haufe, “Synthesis of Vinyl Fluorides by Ring-closing Metathesis”, Tetrahedron Lett. 2004, 45, 57-60.

2003:

G. Haufe, S. Pietz, D. Wölker and R. Fröhlich , "Synthesis of Fluorinated Cycloalkyl N-Phenylcarbamates and Their Microbial Defluorination/Oxygenation by Beauveria bassiana", Eur. J.Org. Chem., 2003, 2166-2175.

G. Haufe and D. Wölker, "Blocking Fluorine Substitution in Biotransformation of Nortricyclanyl N-Phenylcarbamates with Beauveria bassiana", Eur.J. Org. Chem., 2003, 2159-2165.

M. Essers, T. Ernet and G. Haufe, "Enantioselective Diels-Alder reactions of a-fluorinated a,b-unsaturated carbonyl compounds Part 5. Chemical consequences of fluorine substitution", J. Fluorine Chem., 2003, 121, 163-170.

K. Hegemann, H. Schimanski, U. Höweler and G. Haufe, "Selectivity of Candida rugosa Lipase in simultaneous separation of skeletal isomers, desymmetrization and kinetic racemate cleavage of 9-oxabicyclononanediols", Tetrahedron Letters, 2003, 44, 2225-2229.

2002:

M. Essers and G. Haufe, "Chemical Consequences of Fluorine Substitution. Part 4. Diels-Alder Reactions of Fluorinated p-Benzoquinones with Dane's Diene. Synthesis of Fluorinated D-Homosteroids", J. Chem. Soc., Perkin Trans. I, 2002, 2719-2728.

G. Haufe, O. G. J. Meyer and C. Mück-Lichtenfeld, "Addition of Dihalocarbenes to Vinyl Fluorides. Chemical Consequences of Fluorine Substitution. Part 3.", Coll. Czech. Chem. Comm., 2002, 67, 1493-1504.

S. Grimme, A. Bahlmann and G. Haufe, "Ab initio Calculations for the Optical Rotations of Conformationally Flexible Molecules: A Case Study on Six-, Seven- and Eight-membered Fluorinated Cycloalkanol Esters", CHIRALITY 2002, 14, 793-797.

T. C. Rosen and G. Haufe, "Synthesis of Enantiopure, Monofluorinated Phenylcyclopropyl Derivatives by Lipase-catalyzed Kinetic Resolution", Tetrahedron: Asymmetry 2002, 13, 1397-1405.

C. E. Uhlemann, G. Hägele, K. W. Laue, M. Lübke and G. Haufe, "The first ¹⁹F NMR controlled titration. 2-Amino-4-fluoro-2-methylpent-4-enoic acid", Magn. Res. Chem. 2002, 40, 573-580.

M. Essers, C. Mück-Lichtenfeld and G. Haufe, "Diastereoselective Diels-Alder Reactions of a-Fluorinated a,b-Unsaturated Carbonyl Compounds. Chemical consequences of Fluorine Substitution. Part 2.", J. Org. Chem. 2002, 67, 4715-4721.

G. Haufe, T. C. Rosen, O. G. J. Meyer, R. Fröhlich and K. Rissanen, "Synthesis, Reactions and Structural Features of Monofluorinated Cyclopropane Carboxylates", J. Fluorine Chem. 2002, 114, 189.

G. Haufe, D. Wölker and R. Fröhlich, "Selectivity of Biohydroxylation with Beauveria bassiana of trans-2-Fluorocycloalkyl-N-phenylcarbamates", J. Org. Chem. 2002, 67, 3022.

D. Wölker and G. Haufe, "Synthesis of Optically Active Vicinal Fluorohydrins by Lipase-catalyzed Deracemization", J. Org. Chem. 2002, 67, 3015.

G. Haufe and A. Burchardt, "Improved Synthesis of Fluorinated Analogues of Anticancer Active Ether Lipids", Synthesis 2002, 648.

S. Bruns and G. Haufe, "(Salen)chromium Complex Mediated Asymmetric Ring Opening of Meso- and Racemic Epoxides with Different Fluoride Sources", Adv. Synth. Catal. 2002, 344, 165.

M. Fix, S. Wiehle, G. Haufe, and H.-J. Galla, "Synthesis of regioisomeric fluorohydroxylated fatty acid methyl esters and their phase behavior at the air-water interface compared to hydroxylated amphiphiles", Colloids Surfaces A: Physicochem. Engin. Aspects 2002 198-200, 151.

F. Chanteau, M. Essers, R. Plantier-Royon, G. Haufe and C. Portella, "Dienophilic reactivity of perfluoroalkenyl ketones in Diels-Alder reactions", Tetrahedron Lett. 2002, 43, 1677.

2001:

G. Haufe, S. Bruns and M. Runge, "Enantioselective Ring-opening of Epoxides by HF-Reagents. Asymmetric Synthesis of Fluoro Lactones", J. Fluorine Chem. 2001, 112, 55.

G. Haufe and A. Burchardt, "Synthesis of a Fluorinated Ether Lipid Which is Analogous to a Platelet Activating Factor", Eur. J. Org. Chem. 2001, 4501.

M. Essers, B. Wibbeling, G. Haufe, „Synthesis of first fluorinated cantharidin analogues", Tetrahedron Lett. 2001, 42, 5429-5433.

T. Ernet, A. H. Maulitz, E.-U. Würthwein, G. Haufe, „Chemical Consequences of Fluorine Substitution. Part 1. Experimental and Theoretical Results on Diels-Alder Reactions of a- and b-Fluorostyrenes", J. Chem. Soc., Perkin Trans. 1 2001, 1929-1938.

A. Burchardt, T. Takahashi, Y. Takeuchi, G. Haufe, "Synthesis of a-Fluorinated Analogue of Anticancer Active Ether Lipids", J. Org. Chem. 2001, 66, 2078-2084.

2000:

M. Runge, G. Haufe, "Synthesis of a-Fluorinated Analogue of the Antibiotic Lasiodiplodin", J. Org. Chem. 2000, 65, 8737-8742.

O. G. J. Meyer, R. Fröhlich, G. Haufe, „Asymmetric Cyclopropanation of Vinyl Fluorides: Access to Enantiopure Monofluorinated Cyclopropane Carboxylates“, Synthesis 2000, 1479-1490.

K. W. Laue, S. Kröger, E. Wegelius, G. Haufe, „Stereoselective Synthesis of g-Fluorinated a-Amino Acids using 2-Hydroxy-3-pinanone as an Auxiliary“, Eur. J. Org. Chem. 2000, 3737-3743.

W.-R. Abraham, H.-A. Arfmann, K. Kieslich, G. Haufe, „Regioselectivity of the Microbial Hydroxylation of Nortricyclanol and its Derivatives", Biocatalysis & Biotransformation 2000, 18, 283-290.

T. Takahashi, A. Fukushima, Y. Tanaka, M. Segawa, H. Hori, Y. Takeuchi, A. Burchardt, G. Haufe, „New Efficient Derivatizing Agent, a-Cyano-a-fluoro(2-naphthyl)acetic Acid (2-CFNA). Application on the ee Determination of (-)-3-Acetoxy-2-fluoro-2-(hexadecyloxy)propan-1-ol", CHIRALITY 2000, 12, 458-463.

S. Bruns, G. Haufe, „Enantioselective introduction of Fluoride into Organic Compounds. First Asymmetric Ring Opening of Epoxides by Hydrofluorinationg Reagents", J. Fluorine Chem. 2000, 104, 247-254.

V. N. Kovtonyuk, L. S. Kobrina, Yu. V. Gatilov, I.Yu. Bagryanskaya, R. Fröhlich, G. Haufe, „Reactions of Polyfluorinated Cyclohexadienones with Diazoalkanes. I. Formation of Cyclopropanes from Polyfluorinated 2,4-Cyclohexadienones with Diazomethane and Phenyldiazomethane", J. Chem. Soc., Perkin Trans. 1, 2000, 1929-1933.

M. Runge, D. O'Hagan, G. Haufe, „Lipase-catalysed Polymerization of Fluorinated Lactones and Fluorinated Hydroxycarboxylic Acids", J. Polym. Sci. A, Polym. Chem. 2000, 38, 2004-2012.

S.-F. Lu, G. Haufe, K. W. Laue, W. L. Padgett, O. Oshunleti, J. W. Daly, K. L. Kirk, „Syntheses of (R)- and (S)-2- and 6-Fluoronorepinephrine and (R)- and (S)-2- and 6-Fluoro-epinephrine: Effect of Stereochemistry on Fluorine-Induced Adrenergic Selectivities", J. Med. Chem. 2000, 43, 1611-1619.

M. Lübke, R. Skupin, G. Haufe, „Regioselectivity of bromofluorination of functionalized 1-alkenes", J. Fluorine Chem. 2000, 102, 125-135.

F. Tranel, G. Haufe: "Lipase-catalyzed resolution of 2-fluorodecanoic acid", Tetrahedron: Asymmetry 2000, 11, 889-896.

J. Oldendorf, G. Haufe, "Synthesis of g-Fluoro-a,b-unsaturated Carboxylic Esters from Saturated a-Fluoro Aldehydes", J. Prakt. Chem. 2000, 342, 52-57.

K. L. Kirk, B. Jayachandran, B. Herbert, S.-F. Lu, W. L. Padgett, J. W. Daly, G. Haufe, K. W. Laue, "Chemical and Biological Approaches to Non-Racemic Fluorinated Catecholamines and Amino Acids", ACS Symposium Series, Vol 746 , P. V. Ramachandran, Ed., American Chemical Society, Washington, D. C., 2000, pp 194-209.

1999:

S. Bruns, G. Haufe, "Catalytic Asymmetric Ring Opening of Epoxides to Chlorohydrins with Mild Chloride Donors and Enantiopure Titanium Complexes", Tetrahedron: Asymm.1999, 10, 1563-1569.

K. W. Laue, C. Mück-Lichtenfeld, G. Haufe, "Enantioselective Syntheses of 2-Amino-4-fluoropent-4-enoic Acids. Isosteres of Asparagine", Tetrahedron 1999, 55, 10413-10424.

A.A. Bogachev, L.S. Kobrina, O. G. J. Meyer, G, Haufe: "Diels-Alder Reactions of Polyfluorinated 2,4-Cyclohexadienones with a- and b-Fluorostyrenes", J. Fluorine Chem. 1999, 97, 135-143.

S. Otten, R. Fröhlich, G. Haufe, "Synthesis and Structural Characterization of Enantiopure Campher-based Di-, Tri- and Tetrasulfides", Heterocycles 1999, 51, 505-512.

G. Haufe, G. Alvernhe, A. Laurent, T. Ernet, O. Goj, S. Kröger, A. Sattler, "Bromofluorination of Alkenes: 1-Bromo-2-fluoro-2-phenylpropane", Org. Synth. 1999, 76, 159-168.

1998:

S. Otten, R. Fröhlich, G. Haufe, "Synthesis and Structural Characterization of Enantiopure (2R,5R)-(+)-2,5-Dimethyl thiolane", Tetrahedron: Asymmetry 1998, 9, 189-191.

G. Haufe, K. W. Laue, M. U. Triller, Y. Takeuchi, N. Shibata, "Synthesis of g-Fluoro-a-methyl-a-amino Acids. A New Alkylation Procedure for Ester Imines", Tetrahedron 1998, 54, 5929-5938.

K. Hegemann, B. Wibbeling and G. Haufe, "Regioselectivity of Oxysulfenylation of Cycloocta-1,5-diene", J. Prakt. Chem./Chem. Ztg. 1998, 340, 455-458.

Y. Takeuchi, M. Kamezaki, K. Kirihara, G. Haufe, K. W. Laue, N. Shibata, "Chemistry of a-Fluoro-a-amino Acids: The First Synthesis of Fully Protected Dipeptides Containing a-Fluoroglycine", Chem. Pharm. Bull. 1998, 46, 1062-1064.

M. M. Kremlev and G. Haufe, "Halofluorination of 1,2-Difluoro-1,2-di(tolyl)ethene, 1,2,3,4-Tetrafluoro-1,4-di(p-tolyl)butadiene and Its Nonfluorinated Parent Compounds", J. Fluorine Chem. 1998, 90, 121-127.

K. W. Laue, G. Haufe, "2-Fluoroallyl Bromide - A Versatile Fluorinated Building Block. Alkylation of Glycine and Alanine Ester Imines", Synthesis 1998, 1453-1456.

T. Kometani, T. Isobe, M. Goto, Y. Takeuchi, G. Haufe, "Enzymatic Resolution of 2-Fluoro-2-arylacetic Acid Derivatives", J. Mol. Cat. B: Enzymatic 1998, 5, 171-174.

R. Skupin, G. Haufe, "Regioselectivity of the Ring Opening of Propene Oxides Bearing Electron Withdrawing Substituents at the Methyl Group with Olah's Reagent", J. Fluorine Chem. 1998, 92, 155-163.

1997:

W. Bone, C.H. Yeung, R. Skupin, G. Haufe, T.G. Cooper, "Toxicity of Ornidazole and its Analogues to Rat Spermatozoa as Reflected in Motility Parameters", Int. J. Androl. 1997, 20, 347-355.

G. Haufe, "Cyclobutanes by ring contraction", in (A. de Meijere) Houben-Weyl, Methoden der Organischen Chemie, Vol. E17e, 4. Ed., pp 317-367, Thieme-Verlag, Stuttgart, 1997.

G. Haufe, "Cyclobutenes by ring enlargement", in (A. de Meijere) Houben-Weyl, Methoden der Organischen Chemie, Vol. E17f, 4. Ed., pp 697-731, Thieme-Verlag, Stuttgart, 1997.

G. Haufe, "Cyclobutenes by ring contraction", in (A. de Meijere) Houben-Weyl, Methoden der Organischen Chemie, Vol. E17fe, 4. Ed., pp 732-761, Thieme-Verlag, Stuttgart, 1997.

G. Haufe, "Rearrangement Reactions of Cyclobutenes" , in (A. de Meijere) Houben-Weyl, Methoden der Organischen Chemie, Vol. E17f, 4. Ed., pp 875-924, Thieme-Verlag, Stuttgart, 1997.

O. Goj, A. Burchardt, G. Haufe, "A Versatile Approach to Optically Active Primary 2-Fluoro-2-phenylalkanols through Lipase-catalyzed Transformations", Tetrahedron: Asymmetry 1997, 8, 399-408.

A. Sattler, G. Haufe, "Lipase-catalysed enantioselective esterification of b-fluoro-alcohols", Preparative Biotransformations, pp 1:10.70-1:10.76, Wiley, Chichester, 1997.

S. Kröger, G. Haufe, "Synthesis of Racemic g-Fluoro-a-amino acids", Amino Acids 1997, 12, 363372.

S. Kröger, G. Haufe, "Stereoselective Synthesis of some g- and d-Fluoro-a-amino Acids", Liebigs Ann./Recueil 1997, 1201-1206.

R. Skupin, T. G. Cooper, R. Fröhlich, J. Prigge, G. Haufe, "Lipase-Catalyzed resolution of both Enantiomers of Ornidazole and some Analogues", Tetrahedron: Asymmetry 1997, 8, 2453-2464.

T. G. Cooper, C.-H. Yeung, R. Skupin, G. Haufe, "Antifertility Potential of Ornidazole Analogues in Rats", J. Androl. 1997, 18, 431-437.

Th. Ernet, G. Haufe, "Allylic Hydroxylation of Vinyl Fluorides", Synthesis 1997, 953-956.

S. Pietz, R. Fröhlich, G. Haufe, "Microbial Oxygenation of Cycloheptyl-N-phenyl-carbamate and (±)-trans-2-Fluorcycloheptyl-N-phenylcarbamate with Beauveria bassiana", Tetrahedron 1997, 53, 17055-17066.

S. Pietz, D. Wölker, G. Haufe, " Selectivity of the Biooxygenation of N-Phenyl-carbamates by the Fungus Beauveria bassiana", Tetrahedron 1997, 53, 17067-17078.

K. Hegemann, G. Haufe, R. Fröhlich, F. Zippel, "Three 2,5-Disubstituted 9-Oxa-bicyclo[4.2.1]nonanes. Transannular O-Heterocyclization Products of Cycloocta-1,5-diene", Acta Cryst. 1997, C53, 1889-1892.

1996:

G. Haufe, "Triethylamine Trishydrofluoride in Synthesis", J. Prakt. Chem./Chem. Ztg. 1996, 338, 99-113.

G. Haufe, S. Kröger, "Syntheses of g-Fluoro-a-amino Acids", Amino Acids 1996, 11, 409-424.

S. Pietz, G. Haufe, R. Fröhlich, M. Grehl, "Syn-1,5-Dimethylbicyclo[3.2.1]oct-8-yl-N-phenylcarbamate", Acta Cryst. 1996, C52, 469-470.

A. Sattler, G. Haufe, "A Facile Two-Step Synthesis of (omega-1)-Fluoroalkan-omega-olides. Influence of a Vicinal Fluorine Substituent in Nucleophilic Substitutions", Tetrahedron 1996, 52, 5469-5474.

R. H. Janke, G. Haufe, E.-U. Würthwein and J. H. Borkent, "Racemization Barriers of Helicenes. A Computational Study", J. Am. Chem. Soc. 1996, 118, 6031-6035.

O. Goj, G. Haufe, R. Fröhlich, "Structure of 1,3-Dicyclohexyl-2,4-bis(cyclohexyl-imino)1,3-diazetidine: Dimer of Dicyclohexylcarbodiimide", Acta Cryst. 1996, C52, 1554-1556.

O. Goj, G. Haufe, "New Synthetic Routes to 2-Fluoro-2-phenylalkanoic Acids", Liebigs Ann. Chem.1996, 1289-1294.

O. Goj, S. Kotila, G. Haufe, "Convenient Routes to 2-Aryl-2-fluoropropionic acids: First Synthesis of Monofluorinated Analogues of (±)-Ibuprofen, (±)-Naproxen and Related Compounds", Tetrahedron 1996, 52, 12761-12774.

T. Ernet, G. Haufe, "Diels-Alder Reactions of Vinyl Fluorides with 1,3-Diphenyl-isobenzofuran", Tetrahedron Lett. 1996, 37, 7251-7252.

1995:

G. Haufe, U. Weßel, K. Schulze, G. Alvernhe, "Synthesis of Monofluorinated C₄-Building Blocks Based on Methallyl Chloride", J. Fluorine Chem. 1995, 74, 283-291.

A. Sattler, G. Haufe, "Synthesis of (9R)- and (9S)-10-Fluorodecan-9-olide (Fluoro-Phoracantholide I). First Lipase-catalyzed Enantioselective Esterification of b-Fluoroalcohols", Tetrahedron: Asymmetry 1995, 6, 2841-2848.

1994:

L. Weber, R. Hommel, J. Behling, G. Haufe, H. Hennig, "Photocatalytic Oxygenation of Hydrocarbons with (Tetraarylporphyrinato)iron(III) Complexes and Molecular Oxygen. Comparison with Microsomal Cytochrome P-450 Mediated Oxygenation Reactions”, J. Am. Chem. Soc. 1994, 116, 2400.

R. Reinhardt, W. Engewald, O. Goj, G. Haufe, "Enantiomer Separation of Side-Chain Fluorinated Alkylbenzenes by Capillary Gas Chromatography on Cyclodextrin Phases”, Chromatographia 1994, 39, 192.

A. Sattler, G. Haufe, "Synthesis of Fluorinated (±)-Phoracantholide and Related Compounds: Regioselective Access to a Novel Class of Monofluorinated Fatty Acid Derivatives”, Liebigs Ann. Chem. 1994, 921.

H. Poleschner, M. Heydenreich, K. Spindler, G. Haufe "Fluoroselenenylation of Acetylenes with Xenon Difluoride-Diorganyl Diselenide and Xenon Difluoride-Phenylseleno(trialkyl)silanes”, Synthesis 1994, 1043.

A. Sattler, G. Haufe, "High Regioselectivity in the Alternative Cleavage of Terminal Epoxides with Different Sources of Nucleophilic Fluoride”, J. Fluorine Chem. 1994, 69, 185.

C. Saluzzo, A.-M. La Spina, D. Picq, G. Alvernhe, D. Anker, D. Wolf, G. Haufe, "Phénylthio (ou phénylséléno)fluoration d'alcynes par le N-phénylthio (ou le N-phénylséléno) phtalimide associé aux complexes pyridine^.9HF ou Et₃N^.3HF". Bull. Soc. Chim. Fr. 1994, 131, 831.

R. Janke, G. Haufe, "Synthesis of New Penta- and Hexahelicene Dicarboxylates", Zh. Org. Khim. 1994, 30, 1365-1367; Russ. J. Org. Chem. 1994, 30, 1432-1434 (publ. 1995).